SCHEMBL10666182

SCHEMBL10666182

O=C1CCC(c2ccncc2)CC1C(=O)C1CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
AKR1C3 P42330 1/20 0.37
AKR1C1 Q04828 1/20 0.37
PAX8 Q06710 1/20 0.36
MAPT P10636 2/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
ROCK2 O75116 4/20 0.33
CYP19A1 P11511 2/20 0.33
PRKG1 Q13976 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ROCK1 Q13464 3/20 0.33
PKN2 Q16513 3/20 0.33
RPS6KA5 O75582 2/20 0.33
LRRK2 Q5S007 2/20 0.33
TP53 P04637 2/20 0.33
CYP3A4 P08684 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272419 0.84 PDE3B (0.44) PDE3BPDE3AMAPTDDB1CRBN
SCHEMBL10665721 0.83 PDE3B (0.39) PDE3BPDE3AAKR1C3AKR1C1MAPT
SCHEMBL9813079 0.81 PDE3B (0.40) PDE3BPDE3ADDB1CRBNROCK2
SCHEMBL9878558 0.77 KDM4E (0.42) PDE3BPDE3AMAPTCYP19A1ALDH1A1
SCHEMBL26857910 0.70 AKR1C3 (0.50) PDE3BPDE3AAKR1C3AKR1C1PAX8
SCHEMBL14630636 0.69 TLR4 (0.37) ALDH1A1TP53
SCHEMBL785036 0.68 ESR2 (0.59) PDE3BPDE3AMAPTDDB1CRBN
SCHEMBL3988360 0.68 AKR1C3 (0.47) AKR1C3AKR1C1MAPTLMNA
SCHEMBL791422 0.68 MAPK1 (0.41) MAPTALDH1A1TSHR
SCHEMBL10534260 0.68 CYP11B2 (0.45) MAPTALDH1A1CYP3A4TSHRTHPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4782154-A CARDIOTONICS MITSUI TOATSU CHEMICALS, INC. (JP) 1988-11-01 US disclosed