SCHEMBL9814028

SCHEMBL9814028

CCOCCOc1ccc(CCN(CC(O)c2ccccc2)C[C@H](O)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ADRB3 P13945 1/20 0.46
KDM4E B2RXH2 2/20 0.44
BCHE P06276 1/20 0.42
CYP51A1 Q16850 3/20 0.42
KCNH2 Q12809 1/20 0.41
LTB4R Q15722 2/20 0.41
LTB4R2 Q9NPC1 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
LTA4H P09960 1/20 0.41
HTT P42858 1/20 0.41
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9782289 0.87 CYP51A1 (0.57) ADRB3CYP51A1
SCHEMBL9813959 0.87 MEN1 (0.43) MEN1KMT2AADRB3KDM4ECYP51A1
SCHEMBL9813873 0.87 ADRB3 (0.48) MEN1KMT2AADRB3CYP51A1CYP1A2
SCHEMBL9813877 0.87 ADRB3 (0.48) MEN1KMT2AADRB3CYP51A1CYP1A2
SCHEMBL9813880 0.87 ADRB3 (0.48) MEN1KMT2AADRB3CYP51A1CYP1A2
SCHEMBL9782091 0.84 THRA (0.40) MEN1KMT2AADRB3KDM4EBCHE
SCHEMBL9782109 0.80 THRA (0.38) MEN1KMT2AADRB3KDM4EBCHE
SCHEMBL9813947 0.80 MEN1 (0.45) MEN1KMT2AADRB3ALDH1A1TAAR1
SCHEMBL9813906 0.79 ADRB3 (0.45) MEN1KMT2AADRB3CYP1A2CYP2D6
SCHEMBL9782603 0.79 CYP51A1 (0.37) MEN1KMT2AADRB3CYP51A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017619-A Anitdiabetic HOFFMANN-LA ROCHE INC. (US) 1991-05-21 US disclosed