SCHEMBL9782091

SCHEMBL9782091

CCOCCOc1ccc(CCN(CC(O)c2ccccn2)CC(O)c2ccccn2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.40
KCNA5 P22460 2/20 0.38
CYP51A1 Q16850 3/20 0.37
BCHE P06276 1/20 0.37
ADRB3 P13945 1/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
FFAR1 O14842 1/20 0.37
LTB4R Q15722 2/20 0.36
LTB4R2 Q9NPC1 2/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KCNH2 Q12809 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9782109 0.96 THRA (0.38) THRAKCNA5CYP51A1BCHEADRB3
SCHEMBL9782286 0.84 CYP51A1 (0.41) THRACYP51A1ALDH1A1FFAR1HRH3
SCHEMBL9782603 0.84 CYP51A1 (0.37) THRACYP51A1ADRB3ALDH1A1FFAR1
SCHEMBL9814028 0.84 MEN1 (0.48) THRACYP51A1BCHEADRB3ALDH1A1
SCHEMBL9782553 0.82 MAOB (0.42) THRAKCNA5FFAR1
SCHEMBL9782289 0.81 CYP51A1 (0.57) CYP51A1ADRB3
SCHEMBL9782133 0.81 KCNH2 (0.38) THRACYP51A1BCHEADRB3ALDH1A1
SCHEMBL9782152 0.80 ADRB3 (0.54) ADRB3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL9782089 0.79 OPRK1 (0.43) KCNA5CYP51A1BCHEKDM4EKCNH2
SCHEMBL9813873 0.77 ADRB3 (0.48) CYP51A1ADRB3CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988714-A Drugs for treatment of obesity and diabetics, increases protein breakdown, for fattening animals HOFFMANN-LA ROCHE INC. (US) 1991-01-29 US disclosed
US-4800206-A ANTIDIABETIC AGENTS; HYPOGLYCEMIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-01-24 US disclosed