SCHEMBL9814129

SCHEMBL9814129

COc1cc(OC)c2c(c1)C(C#N)CCC2

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.36
HTR1A P08908 1/20 0.36
ATM Q13315 1/20 0.36
ADRA1A P35348 1/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
AR P10275 2/20 0.35
HTR2A P28223 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9814113 0.79 DRD1 (0.39) DRD1ATMADRA1AKMT2AAR
SCHEMBL9814134 0.78 CA1 (0.51) CA1CA2TAS1R3TAS1R1TAS1R2
SCHEMBL8586368 0.75 CHRNA7 (0.47) KMT2AMEN1HTR2A
SCHEMBL9814142 0.74 CHRNA7 (0.44) KMT2AMEN1CA1CA2
SCHEMBL2776134 0.73 HTR2A (0.40) KMT2AMEN1HTR2ACA1CA2
SCHEMBL9814140 0.73 PARP1 (0.49) ADRA1AARCA1CA2
SCHEMBL10751929 0.72 ADRA1A (0.40) ADRA1AARHTR2ACA1CA2
SCHEMBL10752424 0.72 DPP4 (0.32)
SCHEMBL8857004 0.72 ADRA1A (0.43) ADRA1AARCA1CA2
SCHEMBL20478812 0.72 ADRA1A (0.49) ADRA1AAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166937-B1 ADRENERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed
US-4634705-A Adrenergic amidines ABBOTT LABORATORIES (US) 1987-01-06 US disclosed
EP-0166937-A2 Adrenergic compounds ABBOTT LABORATORIES (US) 1986-01-08 EP disclosed