SCHEMBL9817686

SCHEMBL9817686

CCOC(=O)CCCc1ccccc1C#Cc1ccc2c(c1)C(C)(C)CCS2

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RARA P10276 7/20 0.54
RARB P10826 7/20 0.54
RARG P13631 7/20 0.54
CYP3A4 P08684 3/20 0.54
KMT2A Q03164 1/20 0.54
CYP26A1 O43174 1/20 0.45
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
FFAR1 O14842 8/20 0.37
FFAR4 Q5NUL3 5/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RXRA P19793 1/20 0.36
TSPO P30536 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817631 0.97 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817763 0.95 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817659 0.89 RARA (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817673 0.86 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817641 0.85 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817849 0.83 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817773 0.83 RARA (0.55) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817603 0.82 CYP4F2 (0.40) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817722 0.82 RARA (0.63) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817682 0.81 RARA (0.58) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed