SCHEMBL9817682

SCHEMBL9817682

CCOC(=O)CCc1cccc(C#Cc2ccc3c(c2)C(C)(C)CCS3)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RARA P10276 10/20 0.58
RARB P10826 10/20 0.58
RARG P13631 10/20 0.58
CYP3A4 P08684 3/20 0.58
KMT2A Q03164 1/20 0.58
CYP26A1 O43174 2/20 0.48
FFAR1 O14842 5/20 0.39
RXRA P19793 2/20 0.38
CRABP2 P29373 1/20 0.37
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
GRM5 P41594 1/20 0.35
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817641 0.94 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817773 0.94 RARA (0.55) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817758 0.90 RARA (0.62) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817673 0.85 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817763 0.85 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817849 0.85 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817871 0.83 RARA (0.71) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817686 0.81 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817631 0.81 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL10568461 0.81 RARA (0.39) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed