SCHEMBL9817699

SCHEMBL9817699

CCCc1cc2c(cc1C#Cc1ccc(C(CCC)C(=O)OCC)cc1)C(C)(C)CCS2

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.45
RARB P10826 8/20 0.45
RARG P13631 8/20 0.45
CYP3A4 P08684 3/20 0.45
KMT2A Q03164 1/20 0.45
CYP26A1 O43174 2/20 0.37
ACACB O00763 2/20 0.34
CRABP2 P29373 1/20 0.30
RXRA P19793 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817782 0.95 RARB (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817823 0.95 RARB (0.47) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817794 0.94 RARB (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817775 0.93 RARB (0.43) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817829 0.91 RARB (0.47) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817808 0.85 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817691 0.83 RARA (0.47) RARARARBRARGCYP3A4KMT2A
SCHEMBL27314939 0.79 RXRA (0.36) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817738 0.79 RARB (0.55) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817836 0.78 RARB (0.61) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed