SCHEMBL9817801

SCHEMBL9817801

CCCCCSc1cc2c(cc1C#Cc1ccc(C(CCC)C(=O)OCC)cc1)C(C)(C)CCO2

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.34
HNF4A P41235 1/20 0.34
RARB P10826 2/20 0.31
RARG P13631 2/20 0.31
CYP3A4 P08684 1/20 0.30
RARA P10276 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817783 0.99 RXRA (0.34) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817789 0.98 RXRA (0.35) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817708 0.94 RXRA (0.35) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817832 0.93 RXRA (0.36) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817739 0.86 RXRA (0.38) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL27304402 0.86 RXRA (0.35) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817749 0.85 RARB (0.40) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL27314939 0.85 RXRA (0.36) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL27313907 0.85 RXRA (0.38) RXRAHNF4ARARBRARGCYP3A4
SCHEMBL9817643 0.85 CYP26A1 (0.35) RXRAHNF4ARARBRARGCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed