SCHEMBL9817818

SCHEMBL9817818

CCOC(=O)c1cccc(C#Cc2cc3c(cc2C)OCCC3(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 4/20 0.42
RARB P10826 4/20 0.42
RARG P13631 3/20 0.42
KMT2A Q03164 2/20 0.42
CYP3A4 P08684 1/20 0.42
ACACB O00763 1/20 0.42
RXRA P19793 1/20 0.42
HNF4A P41235 1/20 0.42
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPT P10636 2/20 0.36
GRM5 P41594 1/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10571276 0.89 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817666 0.88 RARA (0.49) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817878 0.83 RXRA (0.44) RARARARBRARGKMT2ACYP3A4
SCHEMBL6668066 0.82 RARA (0.57) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817655 0.82 RARA (0.56) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817647 0.80 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817887 0.80 RXRA (0.41) RARARARBRARGKMT2ACYP3A4
SCHEMBL9142284 0.80 RXRA (0.41) RARARARBRARGKMT2ACYP3A4
SCHEMBL9138172 0.80 RXRA (0.41) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817661 0.79 ACACB (0.39) RARARARBRARGKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed