SCHEMBL9817844

SCHEMBL9817844

CCOC(=O)c1ccc(C#Cc2cc3c(cc2SCC)OCCC3(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 9/20 0.44
RARB P10826 9/20 0.44
RARG P13631 6/20 0.44
KMT2A Q03164 3/20 0.44
CYP3A4 P08684 2/20 0.44
RXRA P19793 1/20 0.43
HNF4A P41235 1/20 0.43
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
USP2 O75604 2/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
CYP26A1 O43174 2/20 0.36
CRABP2 P29373 1/20 0.36
CYP26B1 Q9NR63 1/20 0.36
RAB9A P51151 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PRKCG P05129 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817814 0.94 RARB (0.42) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817749 0.90 RARB (0.40) RARARARBRARGKMT2ACYP3A4
SCHEMBL7655159 0.90 KMT2A (0.39) RARARARBRARGKMT2ACYP3A4
SCHEMBL10571276 0.88 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817647 0.87 RARA (0.46) RARARARBRARGKMT2ACYP3A4
SCHEMBL6689600 0.87 RARA (0.54) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817665 0.87 CYP26A1 (0.38) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817663 0.85 RARA (0.44) RARARARBRARGKMT2ACYP3A4
SCHEMBL9180599 0.85 RARA (0.40) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817832 0.84 RXRA (0.36) RARARARBRARGKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed