SCHEMBL9818280

SCHEMBL9818280

CC([C]=O)c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
CYP2C19 P33261 2/20 0.40
CYP2C9 P11712 1/20 0.40
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD11B1 P28845 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL95837 0.83 CYP2C19 (0.35) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL10079991 0.80 HTT (0.40) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL954426 0.78 HTT (0.39) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL1044900 0.77 HTT (0.47) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL910441 0.76 ESR1 (0.46) ALDH1A1GABRA1GABRB2LMNAGAA
SCHEMBL9165861 0.76 ESR1 (0.46) ALDH1A1GABRA1GABRB2LMNAGAA
SCHEMBL11791692 0.74 IDO1 (0.36) HTTCYP2C19CYP2C9ALDH1A1HSD11B1
SCHEMBL2675708 0.74 CYP3A4 (0.38) CYP2C9ALDH1A1CYP3A4ALOX15MAOA
SCHEMBL911040 0.74 GABRA1 (0.58) HTTALDH1A1CYP3A4ALOX15GABRA1
SCHEMBL6141021 0.74 CYP3A4 (0.40) CYP2C9ALDH1A1CYP3A4HSD11B1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126635-B1 NOVEL OXINDOLE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-12-18 EP disclosed
US-4694017-A 2-amido 3(oxindol-3-yl)propionic acids having antiulcer activity OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-09-15 US disclosed
EP-0126635-A2 Novel oxindole derivative OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-11-28 EP disclosed