SCHEMBL9818917

SCHEMBL9818917

N#CC(C(=O)Nc1ccc(Br)cc1)C(=O)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
KMT2A Q03164 8/20 0.48
MEN1 O00255 7/20 0.48
GAA P10253 2/20 0.48
ATM Q13315 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
CNR1 P21554 4/20 0.47
POLB P06746 1/20 0.46
LMNA P02545 4/20 0.46
HTT P42858 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
MAPT P10636 3/20 0.42
TSHR P16473 1/20 0.42
NLRP3 Q96P20 1/20 0.42
S1PR3 Q99500 1/20 0.41
GRIK1 P39086 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819381 1.00 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1GAAATM
SCHEMBL9819202 0.93 KMT2A (0.46) ALDH1A1KMT2AMEN1CNR1LMNA
SCHEMBL9819129 0.93 KMT2A (0.54) ALDH1A1KMT2AMEN1GAAATM
SCHEMBL9819047 0.93 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1GAAATM
SCHEMBL9819100 0.88 MEN1 (0.48) ALDH1A1KMT2AMEN1POLBLMNA
SCHEMBL9818833 0.88 MEN1 (0.48) ALDH1A1KMT2AMEN1POLBLMNA
SCHEMBL9819005 0.88 TP53 (0.50) KMT2AMEN1GAAATMGPR55
SCHEMBL9819133 0.88 TP53 (0.50) KMT2AMEN1GAAATMGPR55
SCHEMBL9819077 0.86 MEN1 (0.48) ALDH1A1KMT2AMEN1GAAATM
SCHEMBL9819392 0.86 CNR1 (0.47) KMT2AMEN1CNR1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed