SCHEMBL9819807

SCHEMBL9819807

O=[N+]([O-])c1cccc(CCCBr)c1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.47
GPR35 Q9HC97 2/20 0.47
ALDH1A1 P00352 5/20 0.43
TDP1 Q9NUW8 3/20 0.41
HPGD P15428 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
S100A4 P26447 1/20 0.36
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690575 0.86 ALDH1A1 (0.58) TSHRALDH1A1TDP1HPGDSIGMAR1
SCHEMBL10977025 0.83 TSHR (0.51) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL1167739 0.82 TSHR (0.53) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL94768 0.81 TSHR (0.52) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL9429301 0.81 ALDH1A1 (0.56) TSHRALDH1A1HPGDSIGMAR1SMN1; SMN2
SCHEMBL27868260 0.81 SIGMAR1 (0.55) TSHRGPR35ALDH1A1SIGMAR1
SCHEMBL14845129 0.81 GPR35 (0.49) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL22614890 0.80 GPR35 (0.47) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL94769 0.79 GPR35 (0.55) TSHRGPR35ALDH1A1TDP1HPGD
SCHEMBL9641198 0.79 TSHR (0.55) TSHRGPR35ALDH1A1TDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4987132-A PLATELET ACTIVATING FACTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-01-22 US disclosed
CN-1030415-A Saturated heterocycle carboxamide derivatives and its preparation method YAMANOUCHI PHARMA CO LTD (JP) 1989-01-18 CN disclosed
EP-0279681-A2 Saturated heterocyclic carboxamide derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1988-08-24 EP disclosed