SCHEMBL9822013

SCHEMBL9822013

OCc1cc(S)n2nccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.40
PRKAA1 Q13131 2/20 0.36
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
KCNN3 Q9UGI6 6/20 0.33
CDK9 P50750 5/20 0.33
CCNT1 O60563 4/20 0.33
CDK2 P24941 3/20 0.33
CCNE1 P24864 2/20 0.33
KCNN1 Q92952 2/20 0.33
KCNN2 Q9H2S1 2/20 0.33
CDK7 P50613 2/20 0.32
CDK13 Q14004 1/20 0.32
CDK12 Q9NYV4 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9822219 0.79 PDE10A (0.40) PDE10APRKAA1PRKAB2PRKAG1PRKAA2
SCHEMBL9301157 0.73 PDE10A (0.43) PDE10AKCNN3CDK9CCNT1
SCHEMBL9822180 0.71 KDM4E (0.37) AURKAKDR
SCHEMBL10579322 0.69 ALDH1A1 (0.40)
SCHEMBL9143480 0.67 GAA (0.43) CDK2CCNE1CDK5
SCHEMBL23529908 0.66 DYRK1A (0.44) CCR1
SCHEMBL12364000 0.66 PDE10A (0.43) PDE10APRKAA1PRKAB2PRKAG1PRKAA2
SCHEMBL9821989 0.66 RECQL (0.35) PDE10A
SCHEMBL7431490 0.66 PRKAB2 (0.54) PDE10APRKAA1PRKAB2PRKAG1PRKAA2
SCHEMBL9822243 0.66 TP53 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4987129-A BACTERICIDES SANKEI PHARMACEUTICAL CO., LTD. (JP) 1991-01-22 US disclosed
US-4958019-A Intermediates for synthesis of cephalosporin compounds SANKEI PHARMACEUTICAL CO., LTD. (JP) 1990-09-18 US disclosed
US-4956462-A Bactericides, ANTIBIOTICS, CEPHALOSPORINS SANKEI PHARMACEUTICAL CO., LTD. (JP) 1990-09-11 US disclosed
EP-0302633-A2 Beta-lactam compound, process for preparing the same, intermediate for synthesis of the same and medicinal composition for bacterially infectious disease therapy containing the same SANKEI PHARMACEUTICAL COMPANY LIMITED (JP) 1989-02-08 EP disclosed