SCHEMBL9822553

SCHEMBL9822553

COC(=O)C1=C[C@@H]2CC[C@@H]3[C@H](CC[C@]4(C)[C@@H]([C@H](C)CO[Si](C)(C)C(C)(C)C)CC[C@@H]34)[C@@]2(C)CC1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.59
SRD5A1 P18405 1/20 0.40
VDR P11473 3/20 0.39
GPBAR1 Q8TDU6 2/20 0.39
CYP2C9 P11712 1/20 0.39
HIF1A Q16665 1/20 0.39
PTPN1 P18031 2/20 0.39
NPC1L1 Q9UHC9 1/20 0.38
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9782796 1.00 SRD5A2 (0.59) SRD5A2SRD5A1VDRGPBAR1CYP2C9
SCHEMBL9782708 0.86 SRD5A2 (0.79) SRD5A2SRD5A1VDRGPBAR1CYP2C9
SCHEMBL10334081 0.86 SRD5A2 (0.79) SRD5A2SRD5A1VDRGPBAR1CYP2C9
SCHEMBL9782700 0.86 SRD5A2 (0.79) SRD5A2SRD5A1VDRGPBAR1CYP2C9
SCHEMBL9348037 0.85 SRD5A2 (0.51) SRD5A2SRD5A1VDRGPBAR1NPC1L1
SCHEMBL9782782 0.84 SRD5A2 (0.46) SRD5A2SRD5A1
SCHEMBL9782776 0.84 SRD5A2 (0.46) SRD5A2SRD5A1
SCHEMBL9348309 0.84 SRD5A2 (0.51) SRD5A2SRD5A1VDRGPBAR1NPC1L1
SCHEMBL11246664 0.82 SRD5A2 (0.48) SRD5A2SRD5A1VDRGPBAR1NPC1L1
SCHEMBL9822544 0.81 SRD5A2 (0.47) SRD5A2SRD5A1VDRGPBAR1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289327-B1 STEROID 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-12-18 EP disclosed
US-4910226-A Estrane compound SMITHKLINE BECKMAN CORPORATION (US) 1990-03-20 US disclosed
EP-0289327-A2 Steroid 5-alpha-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1988-11-02 EP disclosed