SCHEMBL9823071

SCHEMBL9823071

C#CCNc1ccc(S(=O)(=O)N(C)C)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA9 Q16790 1/20 0.65
MMP9 P14780 1/20 0.63
MMP13 P45452 1/20 0.63
ADAM17 P78536 1/20 0.63
LMNA P02545 2/20 0.53
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MAPT P10636 2/20 0.51
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
ABCC9 O60706 1/20 0.42
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500919 0.81 MMP9 (0.76) CA12CA1CA2CA9MMP9
SCHEMBL19252178 0.80 CA2 (0.71) CA12CA1CA2CA9MMP9
SCHEMBL19252182 0.79 CA2 (1.00) CA12CA1CA2CA9MMP9
SCHEMBL30119792 0.79 CA2 (0.69) CA12CA1CA2CA9MMP9
SCHEMBL4029439 0.78 MMP9 (1.00) CA12CA1CA2CA9MMP9
SCHEMBL10430120 0.76 CA12 (0.65) CA12CA1CA2CA9MMP9
SCHEMBL28849819 0.75 LMNA (0.48) CA12CA1CA2CA9MMP9
SCHEMBL10430061 0.75 CA2 (0.63) CA12CA1CA2CA9MMP9
Ammonia Solution, Strong SCHEMBL6695894 0.75 LMNA (0.51) CA12CA1CA2CA9LMNA
SCHEMBL23144665 0.74 MAPT (0.55) LMNAKMT2AKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115003299-A Methods and compounds for restoring function of mutant p53 皮姆维制药公司 2022-09-02 CN disclosed
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed