SCHEMBL9823079

SCHEMBL9823079

C#CCN(Cc1ccc2nc(NC(=O)C(C)(C)C)[nH]c(=O)c2c1)c1ccc(C#N)cc1

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.67
TYMS P04818 6/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823168 0.90 TYMS (0.58) DHFRTYMS
SCHEMBL9300016 0.90 DHFR (0.62) DHFRTYMS
SCHEMBL9823377 0.89 DHFR (0.71) DHFRTYMS
SCHEMBL9823303 0.88 DHFR (0.71) DHFRTYMS
SCHEMBL15912214 0.88 DHFR (0.59) DHFRTYMS
SCHEMBL9823464 0.87 DHFR (0.72) DHFRTYMS
SCHEMBL9823090 0.87 DHFR (0.68) DHFRTYMS
SCHEMBL9823227 0.87 TYMS (0.60) DHFRTYMS
SCHEMBL9299072 0.86 DHFR (0.57) DHFRTYMS
SCHEMBL9823200 0.86 DHFR (0.70) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed