SCHEMBL9823227

SCHEMBL9823227

C#CCN(Cc1ccc2nc(NC(=O)C(C)(C)C)[nH]c(=O)c2c1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TYMS P04818 10/20 0.60
DHFR P00374 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823168 0.90 TYMS (0.58) TYMSDHFR
SCHEMBL9300016 0.88 DHFR (0.62) TYMSDHFR
SCHEMBL9823377 0.87 DHFR (0.71) TYMSDHFR
SCHEMBL9823464 0.87 DHFR (0.72) TYMSDHFR
SCHEMBL9823303 0.87 DHFR (0.71) TYMSDHFR
SCHEMBL9823079 0.87 DHFR (0.67) TYMSDHFR
SCHEMBL9823139 0.86 DHFR (0.55) TYMSDHFR
SCHEMBL15912214 0.86 DHFR (0.59) TYMSDHFR
SCHEMBL9823090 0.85 DHFR (0.68) TYMSDHFR
SCHEMBL9299072 0.85 DHFR (0.57) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed