SCHEMBL9823458

SCHEMBL9823458

CN(C)CCC(=O)c1ccc(C#CCNCc2ccc3nc(NC(=O)C(C)(C)C)[nH]c(=O)c3c2)cc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.33
CTNNB1 P35222 1/20 0.33
TCF7L2 Q9NQB0 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823234 0.92 TYMS (0.33) TYMSMEN1POLBTSHRKMT2A
SCHEMBL9823362 0.90 TYMS (0.33) TYMSMEN1POLBTSHRKMT2A
SCHEMBL9823392 0.88 DHFR (0.40) TYMSMEN1POLBTSHRKMT2A
SCHEMBL9823085 0.85 MMP13 (0.41) CTNNB1TCF7L2MEN1POLBTSHR
SCHEMBL9823173 0.85 CTNNB1 (0.36) TYMSCTNNB1TCF7L2MEN1POLB
SCHEMBL9823207 0.84 DHFR (0.41) TYMSMEN1POLBTSHRKMT2A
SCHEMBL9823096 0.82 DHFR (0.38) MEN1POLBKMT2ASMN1; SMN2
SCHEMBL9823232 0.82 MEN1 (0.36) TYMSMEN1POLBTSHRKMT2A
SCHEMBL9823446 0.79 DHFR (0.56) TYMS
SCHEMBL9823478 0.78 DHFR (0.44) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed