SCHEMBL9824075

SCHEMBL9824075

CN1CCN(c2cc3c(cc2F)c(=O)c2c(=O)[nH]sc2n3-c2ccc(F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
LMNA P02545 2/20 0.52
MEN1 O00255 1/20 0.52
THRB P10828 2/20 0.41
ALDH1A1 P00352 2/20 0.41
DRD3 P35462 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.39
RAD52 P43351 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825198 0.89 LMNA (0.52) KMT2ALMNAMEN1ALDH1A1KDM4E
SCHEMBL9824308 0.83 PRKD3 (0.43)
SCHEMBL8921044 0.81 GAA (0.43) KMT2ALMNAMEN1ALDH1A1DRD3
SCHEMBL9824152 0.81 DRD3 (0.50) KMT2AMEN1ALDH1A1DRD3KDM4E
SCHEMBL9824344 0.81 TNKS (0.39) KMT2ALMNAMEN1
SCHEMBL9824477 0.80 KMT2A (0.55) KMT2ALMNAMEN1THRBALDH1A1
SCHEMBL9824962 0.80 ALK (0.39) KMT2ALMNAMEN1ALDH1A1KDM4E
SCHEMBL607251 0.80
SCHEMBL9824990 0.75
SCHEMBL6807011 0.73 LMNA (0.55) KMT2ALMNAMEN1THRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed