SCHEMBL9824744

SCHEMBL9824744

O=c1[nH]oc2c1c(=O)c1cc(F)c(N3CCNCC3)cc1n2-c1ccc(F)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.55
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 3/20 0.55
HPGD P15428 3/20 0.55
HSD17B10 Q99714 3/20 0.55
CYP2C9 P11712 2/20 0.43
CYP1A2 P05177 1/20 0.43
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
BRD4 O60885 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
CYP2J2 P51589 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDR P35968 2/20 0.37
CYP2C19 P33261 1/20 0.37
THRB P10828 2/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823950 0.90 LMNA (0.46) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824477 0.89 KMT2A (0.55) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9823980 0.87 KDM4E (0.42) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824004 0.84 TOP1 (0.43) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824515 0.84 HPGD (0.35) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824480 0.82 ALDH1A1 (0.38) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL10771643 0.81 LMNA (0.37) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824212 0.81 MEN1 (0.39) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9824887 0.80 ALDH1A1 (0.36) LMNAKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9825198 0.80 LMNA (0.52) LMNAKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed