SCHEMBL9824841

SCHEMBL9824841

CCNCC1CCN(c2nc3c(cc2F)c(=O)c2c(=O)[nH]oc2n3C2CC2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.35
CYP2C9 P11712 2/20 0.35
ATP6V1B2 P21281 1/20 0.35
TBXA2R P21731 1/20 0.35
EDNRA P25101 1/20 0.35
TARBP2 Q15633 1/20 0.35
KMT2A Q03164 1/20 0.33
DPP4 P27487 2/20 0.32
CHRM2 P08172 1/20 0.32
DRD1 P21728 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ABCC4 O15439 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
KCNH2 Q12809 1/20 0.32
CACNA1C Q13936 1/20 0.32
SCN5A Q14524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824074 0.83 KMT2A (0.46) KMT2ADPP4CHRM2
SCHEMBL9824035 0.81 KDM4E (0.39) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9824938 0.81 ALDH1A1 (0.37) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9823975 0.80 CYP2C9 (0.44) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9824452 0.78 DPP4 (0.41) LMNAKMT2ADPP4CHRM2DRD1
SCHEMBL10684474 0.77 KMT2A (0.37) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9437369 0.75 DPP4 (0.57) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9824535 0.74 KMT2A (0.45) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL9647215 0.73 DPP4 (0.47) LMNACYP2C9ATP6V1B2TBXA2REDNRA
SCHEMBL10576703 0.72 IKBKB (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed