SCHEMBL9825591

SCHEMBL9825591

COC1=NOC(CN(C(=O)OC(C)(C)C)C(=O)[C@@H](N)Cc2ccccc2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.36
MLYCD O95822 1/20 0.36
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
ALPI P09923 1/20 0.34
PKM P14618 1/20 0.34
PTGS1 P23219 1/20 0.34
XIAP P98170 1/20 0.34
LMNA P02545 3/20 0.33
JAK2 O60674 1/20 0.33
S1PR4 O95977 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSP90AA1 P07900 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
XBP1 P17861 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KIF11 P52732 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825095 0.89 TGM2 (0.37) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL9826384 0.89 TGM2 (0.37) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL4935929 0.89 TGM2 (0.40) SLC7A5MLYCDITGA4ITGB7ALPI
SCHEMBL9826287 0.88 SLC7A5 (0.37) SLC7A5MLYCDITGA4ITGB7ALPI
SCHEMBL9825696 0.87 SLC7A5 (0.38) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL9825400 0.85 L3MBTL1 (0.33) MLYCDHTTNPSR1MEN1KMT2A
SCHEMBL9825201 0.77 ITGB3 (0.36) ALDH1A1NPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL9825808 0.76 SLC7A5 (0.35) SLC7A5MLYCDITGA4ITGB7ALPI
SCHEMBL4934061 0.76 TGM2 (0.49) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL4934993 0.76 TGM2 (0.49) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237082-B1 3,5-DISUBSTITUTED 4,5-DIHYDROISOXAZOLES AS TRANSGLUTAMINASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1991-05-29 EP disclosed
US-4929630-A SKIN DISORDERS, ACNE, 4,5-DIHYDROISOOXAZOLE PEPTIDES SYNTEX (U.S.A.) INC. (US) 1990-05-29 US disclosed
US-4912120-A Containing amine and amide substitution SYNTEX (U.S.A.) INC. (US) 1990-03-27 US disclosed
EP-0237082-A2 3,5-disubstituted 4,5-dihydroisoxazoles as transglutaminase inhibitors SYNTEX (U.S.A.) INC. (US) 1987-09-16 EP disclosed