SCHEMBL9825960

SCHEMBL9825960

COc1ccc(C(=O)N(CCO)CCO)cc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.64
TSHR P16473 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HSP90AA1 P07900 1/20 0.55
HSP90AB1 P08238 1/20 0.55
BLM P54132 1/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA7 P43166 1/20 0.54
TPMT P51580 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
ACHE P22303 3/20 0.53
ALDH1A1 P00352 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11197542 0.86 ELANE (0.62) ELANETSHRCYP1A2CYP3A4CYP2C9
SCHEMBL13216464 0.83 HSP90AA1 (0.77) ELANETSHRCYP1A2CYP3A4CYP2C9
SCHEMBL7350723 0.82 ACKR3 (0.54) CYP1A2CYP3A4HSP90AA1HSP90AB1BLM
SCHEMBL21498147 0.80 ELANE (0.52) ELANETSHRCYP1A2CYP3A4CYP2C9
SCHEMBL6023472 0.78 CES2 (0.52) TSHRCA1CA2KDM4EHPGD
SCHEMBL6409033 0.78 CYP2C9 (0.66) ELANETSHRCYP1A2CYP3A4CYP2C9
SCHEMBL3893527 0.78 TSHR (0.66) ELANETSHRCYP1A2CYP3A4CYP2C9
SCHEMBL3456951 0.77 ACHE (0.65) ELANETSHRCA12CA1CA2
SCHEMBL27968222 0.77 CYP1A2 (0.52) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7157289 0.76 ALDH1A1 (0.48) CYP3A4ALDH1A1HPGDMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0168003-B1 OXINDOL COMPOUNDS, COMPOSITIONS CONTAINING SAME AND PROCESSES FOR PREPARING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-04-03 EP disclosed
US-4737501-A Substituted piperazinyl oxindol compounds and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-04-12 US disclosed
EP-0168003-A1 Oxindol compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-01-15 EP disclosed
US-4415572-A CARDIOTONIC AND INOTROPIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-15 US disclosed