SCHEMBL9827149

SCHEMBL9827149

CC(CN1CCOC(c2csc(C(F)(F)F)n2)C1)c1ccc(OCCO)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CXCR1 P25024 1/20 0.32
FGFR1 P11362 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
MTOR P42345 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
KCNH2 Q12809 1/20 0.31
DRD2 P14416 3/20 0.30
DRD3 P35462 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9827456 0.94 ALDH1A1 (0.39) ALDH1A1ADRB1ADRB3MEN1KMT2A
SCHEMBL9825690 0.92 ALDH1A1 (0.39) ALDH1A1ADRB1ADRB3MEN1KMT2A
SCHEMBL9825905 0.90 ALDH1A1 (0.38) ALDH1A1ADRB1ADRB3MEN1KMT2A
SCHEMBL9827236 0.90 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AKDM4EHRH3
SCHEMBL9826186 0.90 HRH3 (0.36) ALDH1A1ADRB1ADRB3MEN1KMT2A
SCHEMBL9826520 0.89 CNR2 (0.34) MEN1KMT2AKDM4ETDP1MOGAT2
SCHEMBL9825575 0.88 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL9826243 0.88 ALDH1A1 (0.37) ALDH1A1ADRB1ADRB3MEN1KMT2A
SCHEMBL9827035 0.88 ALDH1A1 (0.37) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL9825436 0.88 PIK3CA (0.35) ALDH1A1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0239815-B1 SUBSTITUTED THIAZOLES AND OXAZOLES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1991-07-24 EP disclosed
EP-0239815-A1 Substituted thiazoles and oxazoles, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-10-07 EP disclosed