SCHEMBL9827558

SCHEMBL9827558

COc1ccc(CCCNCCCC2(O)CCc3cc(OC)c(OC)cc3C2C(C)C)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.43
SLC2A1 P11166 1/20 0.39
KDM4E B2RXH2 3/20 0.38
POLB P06746 2/20 0.38
ABCB1 P08183 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP3A5 P20815 1/20 0.38
ADRB2 P07550 1/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP2D6 P10635 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832224 0.96 SMPD1 (0.43) SMPD1SLC2A1KDM4EPOLBABCB1
SCHEMBL9827619 0.90 ADRB2 (0.39) SMPD1SLC2A1KDM4EABCB1CYP3A4
SCHEMBL9828679 0.89 ADRB2 (0.40) SMPD1KDM4EADRB2ALDH1A1
SCHEMBL9736711 0.86 CYP3A4 (0.45) SMPD1SLC2A1ABCB1CYP3A4CYP3A5
SCHEMBL9827453 0.86 CYP3A4 (0.45) SMPD1SLC2A1ABCB1CYP3A4CYP3A5
Hydrochloric Acid SCHEMBL10793128 0.86 SMPD1 (0.52) SMPD1SLC2A1KDM4EADRB2ALDH1A1
Hydrochloric Acid SCHEMBL10797775 0.86 SMPD1 (0.40) SMPD1SLC2A1KDM4EPOLBABCB1
Hydrochloric Acid SCHEMBL9829237 0.86 CYP3A4 (0.45) SMPD1SLC2A1ABCB1CYP3A4ADRB2
Hydrochloric Acid SCHEMBL9736378 0.86 CYP3A4 (0.45) SMPD1SLC2A1ABCB1CYP3A4ADRB2
Hydrochloric Acid SCHEMBL10792003 0.86 CYP3A4 (0.45) SMPD1SLC2A1ABCB1CYP3A4ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177960-B1 DERIVATIVES OF TETRAHYDRONAPHTHALENE, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOFFMANN LA ROCHE (CH) 1991-03-20 EP disclosed
US-4680310-A HYPOTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1987-07-14 US disclosed
EP-0177960-A2 Derivatives of tetrahydronaphthalene, process and intermediates for their preparation and medicines containing them F. HOFFMANN-LA ROCHE AG (CH) 1986-04-16 EP disclosed