SCHEMBL9827619

SCHEMBL9827619

COCCCOc1cc(CCCNCCC2(O)CCc3cc(OC)c(OC)cc3C2C(C)C)ccc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.39
SMPD1 P17405 1/20 0.39
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
REN P00797 4/20 0.37
SIGMAR1 Q99720 2/20 0.36
CYP3A4 P08684 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP2D6 P10635 1/20 0.35
GAA P10253 1/20 0.34
SLC2A1 P11166 1/20 0.34
ABCB1 P08183 1/20 0.34
CYP3A5 P20815 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828679 0.97 ADRB2 (0.40) ADRB2SMPD1DRD2DRD1DRD4
SCHEMBL9832224 0.93 SMPD1 (0.43) ADRB2SMPD1CYP3A4LMNAKDM4E
SCHEMBL9827558 0.90 SMPD1 (0.43) ADRB2SMPD1CYP3A4LMNAKDM4E
SCHEMBL9827613 0.86 CYP3A4 (0.44) SMPD1DRD2DRD1DRD3REN
SCHEMBL9736711 0.84 CYP3A4 (0.45) ADRB2SMPD1SIGMAR1CYP3A4ALDH1A1
SCHEMBL9827453 0.84 CYP3A4 (0.45) ADRB2SMPD1SIGMAR1CYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL10793128 0.84 SMPD1 (0.52) ADRB2SMPD1DRD2DRD1DRD4
Hydrochloric Acid SCHEMBL9736378 0.83 CYP3A4 (0.45) ADRB2SMPD1SIGMAR1CYP3A4LMNA
Hydrochloric Acid SCHEMBL9829237 0.83 CYP3A4 (0.45) ADRB2SMPD1SIGMAR1CYP3A4LMNA
Hydrochloric Acid SCHEMBL10797775 0.83 SMPD1 (0.40) SMPD1SIGMAR1CYP3A4LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177960-B1 DERIVATIVES OF TETRAHYDRONAPHTHALENE, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOFFMANN LA ROCHE (CH) 1991-03-20 EP disclosed
US-4680310-A HYPOTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1987-07-14 US disclosed