SCHEMBL9828679

SCHEMBL9828679

COCCCOc1ccc(CCCNCCC2(O)CCc3cc(OC)c(OC)cc3C2C(C)C)cc1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.40
DRD2 P14416 5/20 0.40
DRD1 P21728 5/20 0.40
DRD4 P21917 5/20 0.40
DRD3 P35462 5/20 0.40
SMPD1 P17405 1/20 0.37
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
ADRB1 P08588 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
S1PR2 O95136 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
LPAR2 Q9HBW0 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9827619 0.97 ADRB2 (0.39) ADRB2DRD2DRD1DRD4DRD3
SCHEMBL9832224 0.92 SMPD1 (0.43) ADRB2SMPD1KDM4EALDH1A1
SCHEMBL9827558 0.89 SMPD1 (0.43) ADRB2SMPD1KDM4EALDH1A1
SCHEMBL9828675 0.85 CYP3A4 (0.42) DRD2DRD1DRD3SMPD1MEN1
SCHEMBL9827613 0.83 CYP3A4 (0.44) DRD2DRD1DRD3SMPD1MEN1
SCHEMBL9736711 0.83 CYP3A4 (0.45) ADRB2SMPD1ADRB1MEN1KMT2A
SCHEMBL9827453 0.83 CYP3A4 (0.45) ADRB2SMPD1ADRB1MEN1KMT2A
Hydrochloric Acid SCHEMBL10793128 0.82 SMPD1 (0.52) ADRB2DRD2DRD1DRD4DRD3
Hydrochloric Acid SCHEMBL9829237 0.82 CYP3A4 (0.45) ADRB2SMPD1ADRB1MEN1KMT2A
Hydrochloric Acid SCHEMBL10797775 0.82 SMPD1 (0.40) SMPD1KMT2AKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177960-B1 DERIVATIVES OF TETRAHYDRONAPHTHALENE, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOFFMANN LA ROCHE (CH) 1991-03-20 EP disclosed
US-4680310-A HYPOTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1987-07-14 US disclosed