SCHEMBL9828518

SCHEMBL9828518

CC(SSC(C)C1NC(=O)NC1=O)C1NC(=O)NC1=O

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
BACE1 P56817 1/20 0.34
RGS12 O14924 1/20 0.31
PTGER3 P43115 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL498235 0.85 TSHR (0.41) TSHRBACE1
SCHEMBL19604178 0.83 TSHR (0.40) TSHRBACE1
SCHEMBL16597503 0.79 TSHR (0.48) TSHRBACE1RGS12PTGER3
SCHEMBL23596518 0.79 TSHR (0.48) TSHRBACE1RGS12PTGER3
SCHEMBL98976 0.79 TSHR (0.48) TSHRBACE1RGS12PTGER3
SCHEMBL9402162 0.77 TSHR (0.46) TSHRBACE1RGS12PTGER3
SCHEMBL9360332 0.76 TSHR (0.44) TSHRBACE1RGS12PTGER3
SCHEMBL9402143 0.76 TSHR (0.44) TSHRBACE1RGS12PTGER3
SCHEMBL9467064 0.74 TSHR (0.43) TSHRBACE1RGS12PTGER3
SCHEMBL1012467 0.72 KDM4E (0.42) TSHRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298583-B1 AROMATIC THIOETHERS LILLY INDUSTRIES LIMITED (GB) 1991-08-21 EP disclosed
US-4968711-A LEUKOTRIENE ANTAGONISTS LILLY INDUSTRIES LIMITED (GB) 1990-11-06 US disclosed
EP-0298583-A1 Aromatic thioethers LILLY INDUSTRIES LIMITED (GB) 1989-01-11 EP disclosed