SCHEMBL9829994

SCHEMBL9829994

CC(C)(OCc1nc(-c2ccc(Cl)cc2)co1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 13/20 0.49
SLC16A1 P53985 8/20 0.49
MCTS1 Q9ULC4 7/20 0.49
PPARA Q07869 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 1/20 0.41
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
LTA4H P09960 1/20 0.39
KMO O15229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10747798 0.84 LTA4H (0.44) MAPTNPC1RAB9ATDP1L3MBTL1
SCHEMBL9830073 0.78 SLC16A3 (0.55) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9831115 0.75 NOTUM (0.55) SLC16A3SLC16A1MCTS1PPARAMEN1
SCHEMBL9831414 0.75 SMN1; SMN2 (0.56) SLC16A3SLC16A1MCTS1MEN1MAPT
Propionic Acid SCHEMBL10435684 0.75 S1PR1 (0.50) TSHRS1PR1S1PR3LTA4HKMO
SCHEMBL10711669 0.74 LTA4H (0.46) MEN1MAPTKMT2ANPC1RAB9A
Clobuzarit SCHEMBL187456 0.74 SLC16A3 (0.62) SLC16A3SLC16A1MCTS1PPARAMEN1
SCHEMBL9441026 0.73 TSHR (0.58) MAPTTSHRS1PR1S1PR3KMO
SCHEMBL2056285 0.72 S1PR1 (0.51) MEN1CYP1A2CYP3A4CYP2D6MAPT
SCHEMBL9833295 0.72 NOTUM (0.51) MEN1MAPTKMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP claimed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US claimed
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed