SCHEMBL9833295

SCHEMBL9833295

OCc1nc(-c2ccc(Cl)cc2)co1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.51
LTA4H P09960 1/20 0.47
S1PR1 P21453 7/20 0.44
S1PR3 Q99500 2/20 0.44
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
KMO O15229 1/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 2/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9440941 0.83 SIRT2 (0.56) NOTUMLTA4HS1PR1S1PR3SIRT2
SCHEMBL5999162 0.82 S1PR1 (0.42) LTA4HS1PR1ADRB2ADRB1ADRB3
SCHEMBL2056285 0.82 S1PR1 (0.51) NOTUMLTA4HS1PR1S1PR3ADRB2
SCHEMBL203844 0.82 LTA4H (0.47) NOTUMLTA4HS1PR1S1PR3SIRT2
SCHEMBL4142338 0.81 NOTUM (0.49) NOTUMS1PR1ADRB2ADRB1ADRB3
SCHEMBL13732790 0.79 S1PR1 (0.54) LTA4HS1PR1S1PR3MEN1ALDH1A1
SCHEMBL5639322 0.78 ENPP3 (0.59) LTA4HS1PR1S1PR3ADRB2ADRB1
SCHEMBL17887308 0.78 LTA4H (0.44) NOTUMLTA4HS1PR1S1PR3MEN1
SCHEMBL9441026 0.78 TSHR (0.58) S1PR1S1PR3KMOALDH1A1MAPT
SCHEMBL9440535 0.77 LTA4H (0.43) NOTUMLTA4HS1PR1S1PR3SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed