SCHEMBL9830013

SCHEMBL9830013

Cc1oc(-c2ccc(Cl)cc2)nc1COC(C)(C)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 14/20 0.57
PPARG P37231 12/20 0.57
PPARD Q03181 1/20 0.57
HSD17B10 Q99714 1/20 0.54
TARBP2 Q15633 1/20 0.51
SLC16A3 O15427 2/20 0.48
SLC16A1 P53985 2/20 0.48
MCTS1 Q9ULC4 2/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829667 0.88 PPARA (0.57) PPARAPPARGPPARDKDM4E
SCHEMBL9831054 0.86 PPARA (0.55) PPARAPPARGPPARD
SCHEMBL5856261 0.84 PPARA (0.82) PPARAPPARGPPARDHSD17B10TARBP2
SCHEMBL9831297 0.83 SLC16A3 (0.47) PPARAPPARGPPARDHSD17B10TARBP2
Romazarit SCHEMBL43265 0.83 ALDH1A1 (0.50) PPARAPPARGPPARDHSD17B10TARBP2
Romazarit SCHEMBL3226211 0.82 ALDH1A1 (0.49) PPARAPPARGPPARDHSD17B10TARBP2
SCHEMBL11008533 0.78 KDM4E (0.76) PPARAPPARGHSD17B10TARBP2KDM4E
SCHEMBL9830357 0.77 SLC16A3 (0.49) PPARATARBP2SLC16A3SLC16A1MCTS1
SCHEMBL9830073 0.77 SLC16A3 (0.55) PPARAPPARGSLC16A3SLC16A1MCTS1
SCHEMBL9830056 0.76 PPARA (0.50) PPARAPPARGPPARDHSD17B10TARBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP claimed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US claimed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP claimed
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed