SCHEMBL9830357

SCHEMBL9830357

CC(C)(OCc1cnc(-c2ccc(Cl)cc2)o1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 11/20 0.49
SLC16A1 P53985 7/20 0.49
MCTS1 Q9ULC4 7/20 0.49
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
MAP4K4 O95819 4/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
PPARA Q07869 1/20 0.41
PDE5A O76074 1/20 0.41
KCNH2 Q12809 1/20 0.41
MINK1 Q8N4C8 1/20 0.41
TARBP2 Q15633 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10745283 0.84 KDM4E (0.52) KDM4EALDH1A1HPGDMAP4K4CYP1A2
SCHEMBL9831115 0.78 NOTUM (0.55) SLC16A3SLC16A1MCTS1KDM4EALDH1A1
Romazarit SCHEMBL43265 0.77 ALDH1A1 (0.50) SLC16A3SLC16A1MCTS1KDM4EALDH1A1
SCHEMBL9830013 0.77 PPARA (0.57) SLC16A3SLC16A1MCTS1KDM4EPPARA
Romazarit SCHEMBL3226211 0.76 ALDH1A1 (0.49) SLC16A3SLC16A1MCTS1KDM4EALDH1A1
SCHEMBL9831414 0.75 SMN1; SMN2 (0.56) SLC16A3SLC16A1MCTS1ALDH1A1HPGD
SCHEMBL9830073 0.75 SLC16A3 (0.55) SLC16A3SLC16A1MCTS1PPARA
SCHEMBL9831297 0.75 SLC16A3 (0.47) SLC16A3SLC16A1MCTS1ALDH1A1MEN1
Clobuzarit SCHEMBL187456 0.74 SLC16A3 (0.62) SLC16A3SLC16A1MCTS1KDM4EALDH1A1
SCHEMBL9832665 0.72 ALDH1A1 (0.53) KDM4EALDH1A1HPGDMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP claimed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US claimed
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed