SCHEMBL9831297

SCHEMBL9831297

CCc1nc(-c2ccc(Cl)cc2)oc1COC(C)(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 9/20 0.47
SLC16A1 P53985 6/20 0.47
MCTS1 Q9ULC4 5/20 0.47
PPARA Q07869 8/20 0.45
PPARG P37231 6/20 0.45
PPARD Q03181 3/20 0.45
HSD17B10 Q99714 1/20 0.44
TARBP2 Q15633 1/20 0.44
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832364 0.89 HSD17B10 (0.43) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9833217 0.88 HSD17B10 (0.44) PPARAPPARGPPARDHSD17B10TARBP2
Romazarit SCHEMBL43265 0.86 ALDH1A1 (0.50) SLC16A3SLC16A1MCTS1PPARAPPARG
Romazarit SCHEMBL3226211 0.85 ALDH1A1 (0.49) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9830013 0.83 PPARA (0.57) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9830056 0.77 PPARA (0.50) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9832600 0.76 TARBP2 (0.51) PPARAPPARGPPARDHSD17B10TARBP2
SCHEMBL10708196 0.76 PPARD (0.47) SLC16A3SLC16A1MCTS1PPARAPPARG
SCHEMBL9834911 0.76 HSD17B10 (0.48) PPARAHSD17B10TARBP2ALDH1A1LMNA
SCHEMBL10712401 0.75 ALDH1A1 (0.49) PPARAPPARGPPARDHSD17B10TARBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP claimed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US claimed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP claimed
EP-0220573-B1 HETEROCYCLIC COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed
US-4774253-A ETHER,-ACIDS, ESTERS OR AMIDES HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0220573-A1 Heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1987-05-06 EP disclosed