SCHEMBL9830253

SCHEMBL9830253

CCOC(=O)CCNc1cccc(C)c1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.59
GAA P10253 3/20 0.54
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
TOP2A P11388 1/20 0.50
HTT P42858 2/20 0.47
ALDH1A1 P00352 4/20 0.45
MAPT P10636 4/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830404 0.88 MAPT (0.56) NLRP3GAATOP2AHTTALDH1A1
SCHEMBL9830020 0.83 TOP2A (0.61) NLRP3TOP2AALDH1A1HSD17B10USP2
SCHEMBL8115145 0.81 TOP2A (0.53) NLRP3GAACYP3A4CYP2D6TOP2A
SCHEMBL1491077 0.81 NLRP3 (0.70) NLRP3GAACYP3A4CYP2D6HTT
SCHEMBL9829781 0.79 TOP2A (0.51) NLRP3TOP2AHTTALDH1A1MAPT
SCHEMBL9832916 0.79 TOP2A (0.48) NLRP3TOP2AHTTALDH1A1MAPT
SCHEMBL9829339 0.79 MAPT (0.51) NLRP3GAATOP2AHTTALDH1A1
SCHEMBL13737098 0.79 HDAC3 (0.48) NLRP3GAACYP3A4CYP2D6ALDH1A1
SCHEMBL9831014 0.79 TOP2A (0.53) NLRP3GAATOP2AHTTALDH1A1
SCHEMBL9832645 0.79 GAA (0.56) GAATOP2AHTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP disclosed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO disclosed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed