SCHEMBL9830735

SCHEMBL9830735

N#CC(C#N)=C1CCN(c2cccc(Cl)c2)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
MAPT P10636 3/20 0.47
KDM4E B2RXH2 1/20 0.47
HTR1A P08908 2/20 0.45
HTR2A P28223 2/20 0.45
HTR7 P34969 2/20 0.45
HTR6 P50406 2/20 0.45
HTR3E A5X5Y0 2/20 0.45
HTR3B O95264 2/20 0.45
HTR3A P46098 2/20 0.45
HTR3D Q70Z44 2/20 0.45
HTR3C Q8WXA8 2/20 0.45
TP53 P04637 1/20 0.45
CYP1A2 P05177 1/20 0.45
ADRB1 P08588 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
THRB P10828 1/20 0.45
CYP2C9 P11712 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830347 0.85 CHRM2 (0.40) ALDH1A1MAPTKDM4EADRB1
SCHEMBL9832896 0.83 BPTF (0.39) ALDH1A1MAPTHTTLMNAALOX12
SCHEMBL9831038 0.83 ADRB1 (0.45) ALDH1A1MAPTADRB1L3MBTL1CA12
SCHEMBL9831691 0.83 MGLL (0.37) ALDH1A1MAPTTP53L3MBTL1LMNA
SCHEMBL9830313 0.82 MAPT (0.42) ALDH1A1MAPTKDM4EHTR3EHTR3B
SCHEMBL10407528 0.82 MAPT (0.40) ALDH1A1MAPTKDM4EHTR3EHTR3B
SCHEMBL9833011 0.81 CYP1A2 (0.47) ALDH1A1MAPTKDM4ECYP1A2ADRB1
SCHEMBL10408045 0.81 ADRB1 (0.48) ALDH1A1MAPTKDM4ECYP1A2ADRB1
SCHEMBL9830884 0.78 AKR1C3 (0.42) HTTLMNA
SCHEMBL9829774 0.78 MLYCD (0.34) ALDH1A1KDM4EHTR1ATP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP disclosed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO disclosed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed