SCHEMBL9830743

SCHEMBL9830743

COc1cc(Br)cc2c(N(C)C)cc(C)nc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.51
NQO2 P16083 5/20 0.48
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
PRNP P04156 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CRHR1 P34998 5/20 0.36
PDE10A Q9Y233 3/20 0.36
PDE2A O00408 1/20 0.36
PDE5A O76074 1/20 0.36
PDE11A Q9HCR9 1/20 0.36
ERN1 O75460 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829864 0.82 NQO2 (0.50) DHFRNQO2MAPTALDH1A1PRNP
SCHEMBL9830322 0.78 DHFR (0.48) DHFRMAPTALDH1A1CRHR1
SCHEMBL9830058 0.78 NQO2 (0.46) DHFRNQO2MAPTALDH1A1PRNP
SCHEMBL9830239 0.78 NQO2 (0.46) DHFRNQO2MAPTALDH1A1PRNP
SCHEMBL5240783 0.76 DHFR (0.46) DHFRMAPTCRHR1
SCHEMBL20350862 0.69 NQO2 (0.46) DHFRNQO2MAPTALDH1A1PRNP
SCHEMBL22715235 0.69 NQO2 (0.46) NQO2MAPTALDH1A1PRNPNPSR1
SCHEMBL22715357 0.67 NQO2 (0.44) NQO2MAPTALDH1A1PRNPNPSR1
SCHEMBL22750299 0.67 CRHR1 (0.47) NQO2MAPTALDH1A1PRNPNPSR1
SCHEMBL16167165 0.67 NQO2 (0.44) NQO2MAPTALDH1A1PRNPNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed