SCHEMBL9830239

SCHEMBL9830239

COc1cc(Br)cc2c(O)cc(C)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.46
MAPT P10636 2/20 0.41
PRNP P04156 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
APP P05067 2/20 0.38
ERN1 O75460 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
NOD2 Q9HC29 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829864 0.85 NQO2 (0.50) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL20521814 0.82 CYP3A4 (0.44) NQO2MAPTALDH1A1APPERN1
SCHEMBL4757968 0.81 MAPT (0.39) MAPTKMT2ANPC1POLBGAA
SCHEMBL22715235 0.81 NQO2 (0.46) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL9830058 0.81 NQO2 (0.46) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL6590987 0.79 GPR35 (0.51) NQO2ALDH1A1ERN1ALOX15L3MBTL1
SCHEMBL22715357 0.79 NQO2 (0.44) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL9830743 0.78 DHFR (0.51) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL18451103 0.78 LMNA (0.39) NQO2MAPTPRNPNPSR1ALDH1A1
SCHEMBL6080169 0.78 MAPT (0.41) NQO2MAPTALDH1A1APPERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed