SCHEMBL9831023

SCHEMBL9831023

CC1(C)C(=O)Nc2c1cc1c(c2-c2ccccn2)NCN1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.38
PDK4 Q16654 3/20 0.38
ADRA1A P35348 1/20 0.36
EPHX2 P34913 1/20 0.34
PDE3A Q14432 4/20 0.34
PDE4D Q08499 3/20 0.34
PDE5A O76074 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE7A Q13946 1/20 0.34
PDE1C Q14123 1/20 0.34
PGR P06401 4/20 0.34
GSK3B P49841 1/20 0.34
MAT2A P31153 1/20 0.33
MARK3 P27448 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK3 Q15120 1/20 0.33
PDE3B Q13370 3/20 0.33
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10472406 0.82 OPRK1 (0.36) ADRA1APDE3APDE4DPDE5APDE1A
SCHEMBL2268820 0.65 PDK2 (0.50) PDK2PDK4EPHX2PGRGSK3B
SCHEMBL9833639 0.65 ATAD2 (0.47) PDK2PDK4PDE3APDE4DPGR
SCHEMBL31404120 0.65 PDK2 (0.50) PDK2PDK4EPHX2PGRGSK3B
SCHEMBL9559276 0.65 HSD17B10 (0.53) PDK2PDK4PDE3APDE4DPGR
Hydrochloric Acid SCHEMBL30775696 0.64 PDK2 (0.48) PDK2PDK4EPHX2GSK3BMARK3
SCHEMBL12721304 0.60 KDM4E (0.50) PDK2
SCHEMBL24625410 0.60 KDM4E (0.68)
SCHEMBL12721336 0.58 PDK2 (0.48) PDK2
Dipyridyl SCHEMBL28323040 0.57 KDM4E (0.82)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed