SCHEMBL9831258

SCHEMBL9831258

Cc1ccccc1CN1CCC(=C(C#N)C#N)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 4/20 0.48
CYP2A13 Q16696 1/20 0.47
LMNA P02545 3/20 0.46
ACHE P22303 1/20 0.46
CLPP Q16740 1/20 0.43
COMT P21964 1/20 0.43
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 5/20 0.40
MEN1 O00255 3/20 0.40
GAA P10253 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GBA1 P04062 1/20 0.39
PRMT5 O14744 2/20 0.39
WDR77 Q9BQA1 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831957 0.84 COMT (0.46) CYP2C19KMT2ALMNACOMTMAPT
SCHEMBL9831681 0.83 MEN1 (0.49) KMT2AACHECOMTKDM4EALDH1A1
SCHEMBL9832661 0.80 KMT2A (0.52) KMT2AACHEMAPTKDM4EALDH1A1
SCHEMBL9832990 0.77 ALDH1A1 (0.45) KMT2ALMNAKDM4EALDH1A1MEN1
SCHEMBL9831214 0.77 KDM4E (0.50) KMT2AACHEMAPTKDM4EALDH1A1
SCHEMBL9830298 0.76 ALDH1A1 (0.45) KMT2ALMNAACHECLPPMAPT
SCHEMBL14234936 0.73 CYP2C19 (0.67) CYP2C19KMT2ACYP2A13LMNAACHE
SCHEMBL9829461 0.73 CYP2C19 (0.58) CYP2C19KMT2ACYP2A13LMNAACHE
SCHEMBL10408283 0.73 POLB (0.55) KMT2ALMNAMAPTKDM4EALDH1A1
SCHEMBL14939422 0.73 ALDH1A1 (0.50) KMT2ACYP2A13LMNAACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449989-A1 6,7 DIHYDROPYRROLO 3,4-c] PYRIDO 2,3-d] PYRIMIDINE DERIVATIVES Sloan-Kettering Institute For Cancer Research (US) 1991-10-09 EP claimed
WO-1990007496-A1 6,7 DIHYDROPYRROLO[3,4-c] PYRIDO[2,3-d] PYRIMIDINE DERIVATIVES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-07-12 WO claimed
US-4925939-A 6,7-dihydropyrrol[3,4-c]pyrido[2,3-d]pyrimidine derivatives SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-05-15 US disclosed