SCHEMBL9831453

SCHEMBL9831453

Cc1cc(C2Nc3cc4c(cc3N2)C(C)(C)C(=O)N4)ccn1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.38
PDE3B Q13370 11/20 0.38
PDE3A Q14432 11/20 0.38
PDE4A P27815 10/20 0.38
PDE4B Q07343 10/20 0.38
PDE4C Q08493 10/20 0.38
PDE4D Q08499 10/20 0.38
PDK2 Q15119 1/20 0.36
PDK4 Q16654 1/20 0.36
PGR P06401 4/20 0.35
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
BMPR1B O00238 1/20 0.33
BMPR1A P36894 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
ACVR1 Q04771 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10472875 0.85 PGR (0.37) PGRBRD4CREBBP
SCHEMBL9832230 0.85 PGR (0.39) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10471878 0.84 PGR (0.34) PGR
SCHEMBL9832238 0.84 PDE3B (0.36) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL9832061 0.83 PDE3B (0.49) ATAD2PDE3BPDE3APDE4APDE4B
Water SCHEMBL10470996 0.82 PDE3B (0.48) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL9831560 0.82 PGR (0.41) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10566029 0.80 ATAD2 (0.39) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10568435 0.80 ATAD2 (0.41) ATAD2PDE3BPDE3APDE4APDE4B
SCHEMBL10563428 0.79 ATAD2 (0.38) ATAD2PDE3BPDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP claimed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP claimed