SCHEMBL9832064

SCHEMBL9832064

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2ccccc2)c2c1COc1cc(Cl)ccc1-2

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 2/20 0.35
CDK2 P24941 2/20 0.35
CCNA1 P78396 2/20 0.35
RIPK1 Q13546 2/20 0.35
MAPT P10636 3/20 0.35
POLB P06746 1/20 0.35
PTPN1 P18031 1/20 0.35
KCNJ6 P48051 4/20 0.35
KCNJ3 P48549 4/20 0.35
KCNJ5 P48544 3/20 0.35
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
HIF1A Q16665 1/20 0.34
LMNA P02545 1/20 0.34
NR1H4 Q96RI1 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831070 0.93 NR1H4 (0.41) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9831514 0.91 MAPT (0.42) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9832636 0.91 LMNA (0.36) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9834162 0.90 CCNA2 (0.40) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9832438 0.90 MAPT (0.45) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9316748 0.90 MAPT (0.44) CCNA2CDK2CCNA1MAPTPOLB
SCHEMBL9832537 0.90 LMNA (0.42) RIPK1MAPTPOLBKCNJ6KCNJ3
SCHEMBL9833530 0.90 RIPK1 (0.41) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9833393 0.89 ALDH1A1 (0.40) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9834065 0.88 RIPK1 (0.39) CCNA2CDK2CCNA1RIPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed