SCHEMBL9832248

SCHEMBL9832248

CC(C)CC1C(=O)Nc2cc(NC(=O)c3ccncc3)c([N+](=O)[O-])cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.40
GAA P10253 4/20 0.40
ALDH1A1 P00352 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPC1 O15118 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
RAB9A P51151 3/20 0.38
LMNA P02545 3/20 0.38
RECQL P46063 1/20 0.38
PRKAB2 O43741 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
KMT2A Q03164 4/20 0.37
POLB P06746 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833672 0.96 MAPT (0.38) MAPTGAAALDH1A1TDP1NPC1
SCHEMBL11024217 0.93 MAPT (0.48) MAPTGAAALDH1A1NPC1SMN1; SMN2
SCHEMBL9833084 0.89 MAPT (0.51) MAPTGAAALDH1A1NPC1SMN1; SMN2
SCHEMBL9832415 0.85 MAPT (0.51) MAPTGAAALDH1A1NPC1SMN1; SMN2
SCHEMBL9832605 0.85 MAPT (0.42) MAPTGAAALDH1A1TDP1NPC1
SCHEMBL9833492 0.85 MAPT (0.40) MAPTGAAALDH1A1TDP1NPC1
SCHEMBL9833715 0.84 MAPT (0.41) MAPTGAAALDH1A1SMN1; SMN2LMNA
SCHEMBL9833552 0.84 MAPT (0.41) MAPTGAAALDH1A1TDP1NPC1
SCHEMBL9833818 0.82 MAPT (0.42) MAPTGAAALDH1A1TDP1NPC1
SCHEMBL9833059 0.82 HCAR3 (0.40) MAPTGAAALDH1A1TDP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed