SCHEMBL9832273

SCHEMBL9832273

COC(=O)C1C(=O)Nc2cc3[nH]c(-c4ccncc4)nc3cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
GAA P10253 1/20 0.47
ATM Q13315 1/20 0.45
PKN1 Q16512 4/20 0.44
PKN2 Q16513 4/20 0.44
RHEB Q15382 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833477 0.89 PKN1 (0.54) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10372616 0.88 CHEK2 (0.48) PDE3BPDE3AKDM4EALDH1A1HPGD
SCHEMBL9830544 0.88 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9831064 0.88 ALDH1A1 (0.50) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL10470299 0.81 PDE3B (0.55) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834558 0.81 CHRNB2 (0.39) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL10373859 0.79 CHEK2 (0.49) PDE3BPDE3AKDM4EALDH1A1HPGD
SCHEMBL9833942 0.77 KDM4E (0.47) KDM4EALDH1A1HPGDPKN1PKN2
SCHEMBL9833850 0.76 ALDH1A1 (0.53) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL9831067 0.75 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed