SCHEMBL9832697

SCHEMBL9832697

COc1cc(C(=O)C#N)cc(OC)c1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.56
PDE4B Q07343 2/20 0.56
PDE4C Q08493 2/20 0.56
PDE4D Q08499 2/20 0.56
TUBB4A P04350 5/20 0.50
TUBB P07437 5/20 0.50
TUBA3C P0DPH7 5/20 0.50
TUBA1B P68363 5/20 0.50
TUBA4A P68366 5/20 0.50
TUBB4B P68371 5/20 0.50
TUBB3 Q13509 5/20 0.50
TUBB2A Q13885 5/20 0.50
TUBB8 Q3ZCM7 5/20 0.50
TUBA3E Q6PEY2 5/20 0.50
TUBA1A Q71U36 5/20 0.50
TUBA1C Q9BQE3 5/20 0.50
TUBB6 Q9BUF5 5/20 0.50
TUBB2B Q9BVA1 5/20 0.50
TUBB1 Q9H4B7 5/20 0.50
TPMT P51580 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177364 0.81 KMT2A (0.51) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL4797626 0.81 TUBB4A (0.50) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL14216108 0.80 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL11343727 0.80 TSHR (0.48) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL11558866 0.80 TSHR (0.48) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL11348095 0.80 TSHR (0.48) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL976684 0.79 CYP1A2 (0.63) PDE4APDE4BPDE4CPDE4DTPMT
SCHEMBL30413049 0.79 CYP1A2 (0.63) PDE4APDE4BPDE4CPDE4DTPMT
SCHEMBL10429070 0.78 TPMT (0.50) PDE4APDE4BPDE4CPDE4DTUBB4A
SCHEMBL10920836 0.78 ALDH1A1 (0.48) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112321544-B Chiral quaternary carbon cyanide and preparation method thereof 深圳湾实验室坪山生物医药研发转化中心 2023-05-26 CN disclosed
CN-112321544-A Chiral quaternary carbon cyanide and preparation method thereof 深圳湾实验室坪山生物医药研发转化中心 2021-02-05 CN disclosed
EP-0281854-B1 4-CHLORO-OXAZOLES, METHOD FOR THEIR PREPARATION AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1991-12-11 EP disclosed
EP-0281854-A1 4-Chloro-oxazoles, method for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1988-09-14 EP disclosed
US-4371606-A 2-(Halogenomethyl-phenyl)-4-halogeno-oxaxole derivatives, a process for the preparation thereof, and radiation-sensitive compositions containing these derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1983-02-01 US disclosed
EP-0041674-A2 2-(Trichloro-methyl-phenyl)-4-halogen-oxazole derivatives, process for preparing them and radiation-sensitive compositions containing them HOECHST AKTIENGESELLSCHAFT (DE) 1981-12-16 EP disclosed