SCHEMBL9833183

SCHEMBL9833183

CC1(C)C(=O)Nc2cc3c(cc21)NC(C=Cc1ccncc1)N3

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 11/20 0.44
PDE3A Q14432 11/20 0.44
PDE4A P27815 10/20 0.44
PDE4B Q07343 10/20 0.44
PDE4C Q08493 10/20 0.44
PDE4D Q08499 10/20 0.44
ATAD2 Q6PL18 1/20 0.37
PGR P06401 4/20 0.35
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10477799 0.87 PDK2 (0.43) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10373984 0.79 ALDH1A1 (0.40) PDE4B
SCHEMBL9832061 0.79 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9834496 0.78 ATAD2 (0.44) PDE3BPDE3APDE4APDE4BPDE4C
Water SCHEMBL10470996 0.78 PDE3B (0.48) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9833683 0.75 PDE3B (0.46) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9834067 0.75 ATAD2 (0.41) PDE3BPDE3APDE4APDE4BPDE4C
Water SCHEMBL10471047 0.74 PDE3B (0.45) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832387 0.74 ATAD2 (0.45) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9834972 0.73 ATAD2 (0.50) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed