SCHEMBL9833282

SCHEMBL9833282

N#CC(C(=O)Nc1cccc(O)c1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 8/20 0.39
MAPT P10636 5/20 0.37
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
KMT2A Q03164 2/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111901 0.92 TP53 (0.42) TP53MAPTPTGS1PTGS2KMT2A
SCHEMBL9834996 0.91 TP53 (0.38) TP53MAPTALDH1A1TSHRNPSR1
SCHEMBL9833272 0.91 TP53 (0.38) TP53MAPTALDH1A1TSHRNPSR1
SCHEMBL10568020 0.91 POLB (0.42) TP53MAPTALDH1A1TSHRNPSR1
SCHEMBL9316263 0.91 RIPK1 (0.41) TP53MAPTALDH1A1TSHRNPSR1
SCHEMBL9832440 0.91 TP53 (0.40) TP53MAPTTSHRKMT2ARAB9A
SCHEMBL9832144 0.91 RIPK1 (0.41) TP53MAPTALDH1A1TSHRNPSR1
SCHEMBL9833373 0.90 TP53 (0.42) TP53MAPTALDH1A1TSHRRAB9A
SCHEMBL9316246 0.89 IDO1 (0.44) TP53MAPTALDH1A1PTGS1PTGS2
SCHEMBL9831199 0.89 MAPT (0.39) TP53MAPTALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed