SCHEMBL9833576

SCHEMBL9833576

CC(C)CC1C(=O)Nc2cc3[nH]c(-c4ccncc4)nc3cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 3/20 0.44
HSD17B10 Q99714 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RHEB Q15382 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.43
AAK1 Q2M2I8 2/20 0.41
SCD O00767 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11020209 0.92 HPGD (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9831445 0.88 MAPT (0.50) ALDH1A1KDM4EHPGDHSD17B10NPC1
SCHEMBL10470925 0.83 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833204 0.83 RHEB (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10470299 0.82 PDE3B (0.55) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9831067 0.80 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834478 0.80 CHRNB2 (0.40) ALDH1A1KDM4EHPGDHSD17B10RAB9A
SCHEMBL10374413 0.78 PGR (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9830544 0.78 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9559331 0.77 HSD17B10 (0.44) ALDH1A1KDM4EHPGDHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed