SCHEMBL9833707

SCHEMBL9833707

O=C1Cc2cc3nc(-c4ccncc4)[nH]c3cc2N1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.56
PDE3A Q14432 3/20 0.56
PDE4A P27815 1/20 0.54
PDE4B Q07343 1/20 0.54
PDE4C Q08493 1/20 0.54
PDE4D Q08499 1/20 0.54
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 3/20 0.52
HPGD P15428 3/20 0.52
CYP1A2 P05177 2/20 0.52
HSD17B10 Q99714 2/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
RHEB Q15382 1/20 0.52
NPC1 O15118 2/20 0.48
RAB9A P51151 1/20 0.48
SCD O00767 1/20 0.47
PKN1 Q16512 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9833232 0.99 PDE3B (0.55) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9832090 0.85 CYP11B1 (0.62) PDE3BPDE3AALDH1A1KDM4EHPGD
SCHEMBL9382865 0.83 PDE3B (0.56) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9379359 0.78 PDE3B (0.69) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566214 0.77 ALOX5 (0.52) ALDH1A1KDM4EHPGDHSD17B10NPC1
SCHEMBL5618665 0.77 EIF2AK2 (0.38) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10531231 0.76 PDE4A (0.54) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9378683 0.75 PDE4A (0.65) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9834560 0.75 KIF11 (0.41) PDE3BPDE3AALDH1A1KDM4EHPGD
SCHEMBL10697017 0.73 ALDH1A1 (0.49) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed