SCHEMBL9833922

SCHEMBL9833922

CSc1ccn2nc(S(=O)(=O)Nc3c(Cl)cccc3Cl)nc2n1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.34
HSD11B1 P28845 2/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
CCR2 P41597 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.31
THRB P10828 1/20 0.31
HPGD P15428 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358915 0.86 HSD11B1 (0.40) HSD11B1ALDH1A1L3MBTL1TSHRHTR6
SCHEMBL10666553 0.85 TSHR (0.34) HSD11B1TSHR
SCHEMBL9833130 0.81 TSHR (0.34) HSD11B1PKMTSHR
SCHEMBL9831148 0.81 TSHR (0.38) TSHR
SCHEMBL8355239 0.81 HSD11B1 (0.38) KMT2AHSD11B1ALDH1A1L3MBTL1TSHR
SCHEMBL9376842 0.80 GAA (0.32) HSD11B1ALDH1A1TSHRLMNA
SCHEMBL9831903 0.79 TSHR (0.37) HSD11B1ALDH1A1L3MBTL1TSHRHTR6
SCHEMBL9832548 0.79 HTR6 (0.39) HSD11B1TSHRHTR6
SCHEMBL8358876 0.79 TSHR (0.37) HSD11B1ALDH1A1L3MBTL1TSHRHTR6
SCHEMBL8355273 0.79 SMN1; SMN2 (0.41) KMT2AMEN1ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
US-4954163-A PRE-AND POSTEMERGENCE HERBICIDES THE DOW CHEMICAL COMPANY (US) 1990-09-04 US disclosed
US-4886883-A HERBICIDES THE DOW CHEMICAL COMPANY (US) 1989-12-12 US disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed